- They are protein in nature and found at the different sites in the cell.
- Drug must interact with the receptor to be able to produce effect.
- The drug receptor complex is similar to the relationship between a lock-and-key theory. Drug should be structurally compatible to the receptors or vice versa.
- A single receptor can react with a number of drugs if the drug conforms to the receptor.
- The intensity of the drug to mediate a response must be proportional to the number of receptors occupied by the drug.
- Drugs attached to the receptors can be classified as an agonist or antagonist.